https://nova.newcastle.edu.au/vital/access/manager/Index ${session.getAttribute("locale")} 5 Pyrimidine-based inhibitors of dynamin I GTPase activity: competitive inhibition at the pleckstrin homology domain https://nova.newcastle.edu.au/vital/access/manager/Repository/uon:32119 (CME) = 65.9 ± 7.7 to 3.7 ± 1.1 mM), which makes this series among the more potent inhibitors of dynamin and CME yet reported. In CME and growth inhibition cell-based assays, the data obtained was consistent with dynamin inhibition. CEREP ExpresS profiling identified off-target effects at the cholecystokinin, dopamine D₂, histamine H₁ and H₂, melanocortin, melatonin, muscarinic M₁ and M₃, neurokinin, opioid KOP and serotonin receptors.]]> Thu 03 May 2018 12:18:53 AEST ]]> Inhibition of dynamin mediated endocytosis by the dynoles-synthesis and functional activity of a family of indoles https://nova.newcastle.edu.au/vital/access/manager/Repository/uon:8338 Sat 24 Mar 2018 08:37:03 AEDT ]]> The antiplasmodial activity of norcantharidin analogs https://nova.newcastle.edu.au/vital/access/manager/Repository/uon:9348 Sat 24 Mar 2018 08:36:28 AEDT ]]> Parallel solution-phase synthesis of targeted tyrphostin libraries with anticancer activity https://nova.newcastle.edu.au/vital/access/manager/Repository/uon:1723 Sat 24 Mar 2018 08:27:23 AEDT ]]> An Ugi-intramolecular Diels-Alder route to highly substituted tetrahydroepoxyisoindole carboxamides https://nova.newcastle.edu.au/vital/access/manager/Repository/uon:12523 Sat 24 Mar 2018 08:16:01 AEDT ]]> Iminochromene inhibitors of Dynamins I and II GTPase activity and Endocytosis https://nova.newcastle.edu.au/vital/access/manager/Repository/uon:11334 Sat 24 Mar 2018 08:13:29 AEDT ]]> A novel class of anticancer compounds targets the actin cytoskeleton in tumor cells https://nova.newcastle.edu.au/vital/access/manager/Repository/uon:19635 Sat 24 Mar 2018 08:01:14 AEDT ]]> Pyrimidyn compounds: dual-action small molecule pyrimidine-based dynamin inhibitors https://nova.newcastle.edu.au/vital/access/manager/Repository/uon:19893 Sat 24 Mar 2018 07:57:02 AEDT ]]> Norcantharidin analogues: synthesis, anticancer activity and protein phosphatase 1 and 2A inhibition https://nova.newcastle.edu.au/vital/access/manager/Repository/uon:5130 Sat 24 Mar 2018 07:48:56 AEDT ]]> BiCl3-mediated opening of epoxides, a facile route to chlorohydrins or amino alcohols: one reagent, two paths https://nova.newcastle.edu.au/vital/access/manager/Repository/uon:341 Sat 24 Mar 2018 07:42:27 AEDT ]]> Norcantharimides, synthesis and anticancer activity: synthesis of new norcantharidin analogues and their anticancer evaluation https://nova.newcastle.edu.au/vital/access/manager/Repository/uon:3264 Sat 24 Mar 2018 07:21:22 AEDT ]]> Synthesis and biological evaluation of norcantharidin analogues: towards PP1 selectivity https://nova.newcastle.edu.au/vital/access/manager/Repository/uon:3263 Sat 24 Mar 2018 07:21:22 AEDT ]]> Long chain amines and long chain ammonium salts as novel inhibitors of dynamin GTPase activity https://nova.newcastle.edu.au/vital/access/manager/Repository/uon:3266 Sat 24 Mar 2018 07:21:22 AEDT ]]> Heterocyclic substituted cantharidin and norcantharidin analogues-synthesis, protein phosphatase (1 and 2A) inhibition, and anti-cancer activity https://nova.newcastle.edu.au/vital/access/manager/Repository/uon:3265 Sat 24 Mar 2018 07:21:21 AEDT ]]>